Rh(III)-Catalyzed C-H Amidation of Indoles with Isocyanates.

نویسندگان

  • Taejoo Jeong
  • Sangil Han
  • Neeraj Kumar Mishra
  • Satyasheel Sharma
  • Seok-Yong Lee
  • Joa Sub Oh
  • Jong Hwan Kwak
  • Young Hoon Jung
  • In Su Kim
چکیده

The rhodium(III)-catalyzed direct amidation of indoles and pyrroles with aryl and alkyl isocyanates is described. These transformations provide a facile and efficient construction of C2-amidated N-heterocyclic scaffolds.

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Rh(III)-catalyzed directed C–H bond amidation of ferrocenes with isocyanates

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عنوان ژورنال:
  • The Journal of organic chemistry

دوره 80 14  شماره 

صفحات  -

تاریخ انتشار 2015